Elenbecestat
CAS No. : 1388651-30-6
(Synonyms: E2609)
| Size | Price | Stock |
|---|---|---|
| 5mg | $190 | In-stock |
| 10mg | $320 | In-stock |
| 25mg | $660 | In-stock |
| 50mg | $1100 | In-stock |
| 100mg | $1700 | In-stock |
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| 500 mg | Get quote | |
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| Cat. No. : | HY-109055 |
| M.Wt: | 437.44 |
| Formula: | C19H18F3N5O2S |
| Purity: | >98 % |
| Solubility: | DMSO : 100 mg/mL (ultrasonic) |
Elenbecestat (E2609) is a potent, orally bioavailable and BBB-penetrant BACE-1 inhibitor. Elenbecestat has the potential for Alzheimer's disease (AD) research[1][2].
IC50 & Target:BACE-1[1]
In Vitro:Elenbecestat (E2609) is a potent BACE1 inhibitor with an IC50 of ~7 nmol/L in cell-based assay[2].
Elenbecestat has been shown to reduce Ab production in the plasma, brain, and cerebrospinal fluid (CSF) of rodents[2].
In Vivo:Elenbecestat (E2609; 0.3-30 mg/kg; p.o.) potently inhibits Ab1-40 and Ab1-42 production in the plasma and CSF of non-human primates[2].
Elenbecestat displays the plasma half-life of 12-16 hours after once daily dosing[1].
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