LY2795050
CAS No. : 1346133-08-1
| Size | Price | Stock |
|---|---|---|
| 5mg | $190 | In-stock |
| 10mg | $310 | In-stock |
| 50mg | $740 | In-stock |
| 100mg | $1100 | In-stock |
| 200 mg | Get quote | |
| 500 mg | Get quote | |
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| Cat. No. : | HY-15708 |
| M.Wt: | 407.89 |
| Formula: | C23H22ClN3O2 |
| Purity: | >98 % |
| Solubility: | DMSO : 50 mg/mL (ultrasonic) |
LY2795050 is a short-acting selective κ(kappa)-opioid receptor (KOR) antagonist. LY2795050 has high affinity for the KOR with Ki value of 0.72 nM. LY2795050 can be used for the research of central nervous system dysfunction[1][2].
IC50 & Target: Ki: 0.72 nM (KOR); Kb: 0.63 nM (KOR)[1]
In Vitro: LY2795050 displays high affinity with a Ki value of 0.72 nM for the KOR and has antagonist activity with a Kb value of 0.63 nM[1].
In Vivo: LY2795050 (i.p., 0.032-0.1mg/kg, 30 min) prevents dose-dependent grooming deficits produced by U50,488 in male and female mice[2].
LY2795050 (i.p., 0.032-0.1mg/kg, 0-150 min) has sexual dimorphism in some behavioral effects[2].
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