XMD16-5
CAS No. : 1345098-78-3
| Size | Price | Stock |
|---|---|---|
| 5mg | $120 | In-stock |
| 10mg | $180 | In-stock |
| 25mg | $288 | In-stock |
| 50mg | $528 | In-stock |
| 100mg | $960 | In-stock |
| 200 mg | Get quote | |
| 500 mg | Get quote | |
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| Cat. No. : | HY-101243 |
| M.Wt: | 416.48 |
| Formula: | C23H24N6O2 |
| Purity: | >98 % |
| Solubility: | DMSO : 100 mg/mL (240.11 mM; Need ultrasonic) |
XMD16-5 is a potent TNK2 inhibitor with IC50 values of 16 and 77 nM for the D163E and R806Q mutations, respectively. IC50 & Target: IC50: 16 nM (TNK2, D163E mutation), 77 nM (TNK2, R806Q mutation)[1] In Vitro: XMD16-5 potently inhibits the growth of the TNK2 mutant expressing cell lines while having little or no effect on the control cells out to the highest tested concentrations (1,000 nM). XMD16-5 has IC50s of 16 nM and 77 nM for the D163E and R806Q mutations. The effects of XMD16-5 on TNK2 cell lines are largely due to on-target effects on TNK2. Auto-phosphorylation of overexpressed TNK2 mutants could be blocked with TNK2 inhibitor XMD16-5[1].
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Inquiry Information- Product Name:
- XMD16-5
- Cat. No.:
- HY-101243
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