VU0360172
CAS No. : 1310012-12-4
| Size | Price | Stock |
|---|---|---|
| 5mg | $150 | In-stock |
| 10mg | $240 | In-stock |
| 25mg | $480 | In-stock |
| 50mg | $750 | In-stock |
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| 200 mg | Get quote | |
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| Cat. No. : | HY-120589 |
| M.Wt: | 294.32 |
| Formula: | C18H15FN2O |
| Purity: | >98 % |
| Solubility: | DMSO : 83.33 mg/mL (ultrasonic) |
VU0360172 is a potent and selective mGlu5 receptor positive allosteric modulator with an EC50 value of 16 nM and a Ki of 195 nM, respectively. VU0360172 stimulates polyphosphoinositide (PI) hydrolysis in vivo, which is abrogated in mGlu5 receptors gene deleted mice[1]. VU0360172 is a click chemistry reagent, itcontains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.
IC50 & Target:EC50: 16 nM (mGlu5 receptor)[1]
Ki: 195 nM (mGlu5 receptor)[1]
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