LY2940094 (tartrate)
CAS No. : 1307245-87-9
(Synonyms: BTRX-246040 (tartrate))
| Size | Price | Stock |
|---|---|---|
| 5mg | $220 | In-stock |
| 10mg | $385 | In-stock |
| 25mg | $770 | In-stock |
| 50mg | $1078 | In-stock |
| 100 mg | Get quote | |
| 200 mg | Get quote | |
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| Cat. No. : | HY-114452A |
| M.Wt: | 631.05 |
| Formula: | C26H29ClF2N4O8S |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
LY2940094 (BTRX-246040) tartrate is a potent, brain penetrant, selective and orally available N/OFQ peptide (NOP) receptor antagonist with high affinity (Ki=0.105 nM) and antagonist potency (Kb=0.166 nM). LY2940094 tartrate reduces Ethanol self-administration and Ethanol seeking in animal models[1].
IC50 & Target: Ki: 0.105 nM (NOP receptor)[1]
Kb: 0.166 nM (NOP receptor)[1]
In Vivo: LY2940094 (3, 10, or 30 mg/kg; orally daily for 4 days) dose-dependently reduces homecage ethanol self-administration in Indiana Alcohol-Preferring (P) and Marchigian Sardinian Alcohol-Preferring (msP) rats, without affecting food/water intake or locomotor activity[1].
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