Darolutamide (Standard)
CAS No. : 1297538-32-9
(Synonyms: ODM-201 (Standard); BAY-1841788 (Standard))
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| Cat. No. : | HY-16985R |
| M.Wt: | 398.85 |
| Formula: | C19H19ClN6O2 |
| Purity: | >98 % |
| Solubility: |
Darolutamide (Standard) is the analytical standard of Darolutamide (HY-16985). This product is intended for research and analytical applications. Darolutamide (ODM-201) is an orally active competitive androgen receptor (AR) antagonist, with a Ki of 11 nM for rat wild-type AR (wtAR) and an IC50 of 26 nM for human wild-type AR (hAR)-mediated transcriptional activation[1]. Darolutamide inhibits testosterone-induced AR nuclear translocation and transcriptional activation[1]. Darolutamide exerts selective effects on AR-positive cells by inhibiting AR-dependent signaling pathways, and its active metabolite retains full antagonistic activity against AR mutants[1]. Darolutamide can be used for the research of prostate cancer, including androgen receptor-dependent prostate cancer[1]. IC50 & Target:IC50: 26 nM (AR-HEK293 cells, AR)[1]
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