Dehydroaripiprazole
CAS No. : 129722-25-4
(Synonyms: OPC-14857; DM-14857)
| Size | Price | Stock |
|---|---|---|
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| 250mg | $205 | In-stock |
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| Cat. No. : | HY-100665 |
| M.Wt: | 446.37 |
| Formula: | C23H25Cl2N3O2 |
| Purity: | >98 % |
| Solubility: | DMSO : 20 mg/mL (ultrasonic;warming;heat to 60°C) |
Dehydroaripiprazole (OPC-14857) is an active metabolite of Aripiprazole (HY-14546) and dopamine D2/D3 receptor partial agonist. Dehydroaripiprazole also has certain affinity for serotonin 5-HT1A, 5-HT2A and 5-HT2B receptors. Dehydroaripiprazole has antipsychotic activity equivalent to Aripiprazole[1][2][3][4][5][6][7][8].
IC50 & Target:5-HT2A and 5-HT2B
In Vitro:Dehydroaripiprazole (0.1-30 μM; 5 min) shows a concentration-dependent inhibitory effect on BCRP-mediated [3H]-MTX uptake in BCRP-expressing membrane vesicles, with an IC50 value of 0.52 μM[5].
Dehydroaripiprazole acts as a dopamine D2/D3 receptor partial agonist in Chinese hamster ovary (CHO) cell[6].
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