TBK1/IKKε-IN-2
CAS No. : 1292310-49-6
| Size | Price | Stock |
|---|---|---|
| 5mg | $250 | In-stock |
| 10mg | $390 | In-stock |
| 25mg | $620 | In-stock |
| 50mg | $840 | In-stock |
| 100mg | $1100 | In-stock |
| 200 mg | Get quote | |
| 500 mg | Get quote | |
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| Cat. No. : | HY-12453 |
| M.Wt: | 457.52 |
| Formula: | C26H27N5O3 |
| Purity: | >98 % |
| Solubility: | DMSO : 21.5 mg/mL (ultrasonic;warming) |
TBK1/IKKε-IN-2 is a dual TBK1 and IKKε inhibitor. IC50 & Target: IC50: 0.6 nM (TBK1, at 5 μM ATP), 2.6 nM (TBK1, at 250 μM ATP), 3.9 nM (IKKε, at 10 μM ATP)[1] In Vitro: TBK1/IKKε-IN-2 (Cmpound #1) inhibits TBK1 biochemical function in Ulight kinase assay at 5 and 250 μM ATP concentration with IC50s of 0.6 and 2.6 nM, rsespectively. TBK1/IKKε-IN-2 inhibits IKKε biochemical function in Ulight kinase assay at 10 μM ATP with an IC50 of 3.9 nM. The IC50 of TBK1/IKKε-IN-2 in the Panc 02.13 proliferation assay is 5 μM[1].
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- TBK1/IKKε-IN-2
- Cat. No.:
- HY-12453
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