KB-5492 (anhydrous)
CAS No. : 129200-10-8
| Size | Price | Stock |
|---|---|---|
| 5mg | $430 | In-stock |
| 10mg | $700 | In-stock |
| 25mg | $1400 | In-stock |
| 50mg | $2300 | In-stock |
| 100mg | $3700 | In-stock |
| 200 mg | Get quote | |
| 500 mg | Get quote | |
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| Cat. No. : | HY-19120 |
| M.Wt: | 546.57 |
| Formula: | C27H34N2O10 |
| Purity: | >98 % |
| Solubility: | DMSO : 250 mg/mL (ultrasonic);DMSO : 250 mg/mL (ultrasonic) |
KB-5492 anhydrous is a potent and selective inhibitor of sigma receptor, inhibits specific [3H]1,3-di(2-tolyl)guanidine (DTG) binding to the sigma receptor with an IC50 of 3.15 μM. KB-5492 anhydrous is an anti-ulcer agent[1][2].
IC50 & Target: IC50: 3.15 μM (sigma receptor)[1]
In Vitro: KB-5492 (0.001-100 μM) inhibits specific [3H]DTG binding in a concentration-dependent manner[1].
KB-5492 (0.1-1 mM) significantly and concentration-dependently prevents the ethanol- and acidified aspirin-induced increases in 51Cr release from gastric epithelial cells[2].
In Vivo: KB-5492 (200?mg/kg; p.o.) prevents macroscopic lesions in the gastric mucosa[2].
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Inquiry Information- Product Name:
- KB-5492 (anhydrous)
- Cat. No.:
- HY-19120
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