(1R,2R)-2-PCCA


CAS No. : 1287205-42-8

1287205-42-8
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Cat. No. : HY-100013A
M.Wt: 455.63
Formula: C30H37N3O
Purity: >98 %
Storage: at 20℃ 2 years
Solubility: DMSO
Introduction of 1287205-42-8 :

(1R,2R)-2-PCCA is a diastereomer of 2-PCCA, and acts as a potent GPR88 receptor agonist, with an EC50 of 3 nM. IC50 & Target: EC50: 3 nM (GPR88 receptor)[1] In Vitro: (1R,2R)-2-PCCA (Example 3) is a potent GPR88 receptor agonist, with an EC50 of 3 nM[1]. (1R,2R)-2-PCCA inhibits GPR88-mediated cAMP production through a Gαi-coupled pathway, with an EC50 of 56 nM in HEK293 cells stably expressing the human GPR88 receptor and the GloSensor-22F cAMP construct[2].

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