Enarodustat
CAS No. : 1262132-81-9
(Synonyms: JTZ-951; SAL0951)
| Size | Price | Stock |
|---|---|---|
| 5mg | $94 | In-stock |
| 10mg | $154 | In-stock |
| 50mg | $440 | In-stock |
| 100mg | $825 | In-stock |
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| Cat. No. : | HY-109057 |
| M.Wt: | 340.33 |
| Formula: | C17H16N4O4 |
| Purity: | >98 % |
| Solubility: | DMSO : 83.33 mg/mL (ultrasonic) |
Enarodustat is a potent and orally active hypoxia-inducible factor prolyl hydroxylase inhibitor, with an EC50 of 0.22 μM. Enarodustat has the potential for renal anemia treatment. IC50 & Target:EC50: 0.22 μM (factor prolyl hydroxylase)[1] In Vitro: Enarodustat (JTZ-951) is a potent and orally active hypoxia-inducible factor prolyl hydroxylase inhibitor, with an EC50 of 0.22 μM. Enarodustat exhibits neither CYP (IC50 > 100 μM; CYP3A4/5, CYP2C9, CYP2D6, CYP1A2, CYP2A6, CYP2C19, CYP2C8, CYP2B6) nor hERG (IC50 > 100 μM) inhibition[1]. In Vivo: Enarodustat (1 and 3 mg/kg, p.o.) increases hemoglobin levels in a dose-dependent manner with daily oral dosing in rats[1].
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