Tipelukast
CAS No. : 125961-82-2
(Synonyms: KCA 757; MN 001)
| Size | Price | Stock |
|---|---|---|
| 1mg | $200 | In-stock |
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| Cat. No. : | HY-14938 |
| M.Wt: | 530.67 |
| Formula: | C29H38O7S |
| Purity: | >98 % |
| Solubility: | Ethanol : 1 mg/mL (ultrasonic;warming) |
Tipelukast (KCA 757) is a sulfidopeptide leukotriene receptor antagonist, an orally bioavailable anti-inflammatory agent and used for the treatment of asthma. In Vitro: Tipelukast inhibits the binding of [3H] LTD4 to the LTD4 receptors on pul-monary cell membrane of guinea-pigs (IC50 = 2.3 μmol)[2]. In Vivo: Fiftheen min after an aerosolized antigen challenge, and UNDW inhaled 5 min later into the guinea pigs, Tipelukast significantly alters the UNDW-induced bronchoconstriction[1]. Tipelukast (1 and 5 mg/kg) administered intravenously 15 min after antigen challenge reduces the propranolol-induced bronchoconstriction (PIB) in a dose-dependent manner in guinea-pigs[2].
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