GNE-0439
CAS No. : 1241902-40-8
| Size | Price | Stock |
|---|---|---|
| 5mg | $500 | In-stock |
| 10mg | $850 | In-stock |
| 25mg | $1750 | In-stock |
| 50mg | $2800 | In-stock |
| 100mg | $4500 | In-stock |
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| Cat. No. : | HY-123824 |
| M.Wt: | 345.48 |
| Formula: | C21H31NO3 |
| Purity: | >98 % |
| Solubility: | DMSO : 130 mg/mL (ultrasonic) |
GNE-0439 is a novel Nav1.7-selective inhibitor with IC50 of 0.34 uM and inhibits Nav1.5 with an IC50 of 38.3 μM. GNE-0439 inhibits mutant N1742K channels (IC50=0.37 uM) in membrane potential assays. GNE-0439 possesses a carboxylic acid group, binds outside of the channel pore, and is unique compared with known selective VSD4 binders[1]. IC50 & Target: IC50: 0.34 uM (Nav1.7)[1]
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