PF-05186462
CAS No. : 1235406-03-7
| Size | Price | Stock |
|---|---|---|
| 5mg | $360 | In-stock |
| 10mg | $540 | In-stock |
| 25mg | $900 | In-stock |
| 50mg | $1260 | In-stock |
| 100mg | $2105 | In-stock |
| 200 mg | Get quote | |
| 500 mg | Get quote | |
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| Cat. No. : | HY-122001 |
| M.Wt: | 531.89 |
| Formula: | C19H10ClF4N5O3S2 |
| Purity: | >98 % |
| Solubility: | DMSO : 50 mg/mL (ultrasonic) |
PF-05186462 is a potent and selective inhibitor of human Nav1.7 voltage-dependent sodium channel, with an IC50 of 21 nM. PF-05186462 shows significant selectivity for Nav1.7 versus other sodium channels (Nav 1.1, 1.2, 1.3, 1.4, 1.5, 1.6, and 1.8). PF-05186462 can be used for the research of acute or chronic pain[1].
IC50 & Target:IC50: 21 nM (human Nav1.7)[1]
In Vitro:PF-05186462 inhibits human Nav1.7 channels (IC50=21 nM) in HEK293 cells[1].
PF-05186462 exhibits a high plasma protein binding rate[1].
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