Azelnidipine
CAS No. : 123524-52-7
(Synonyms: CS 905)
| Size | Price | Stock |
|---|---|---|
| 5mg | $55 | In-stock |
| 10mg | $77 | In-stock |
| 25mg | $138 | In-stock |
| 50mg | $220 | In-stock |
| 100mg | $350 | In-stock |
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| Cat. No. : | HY-B0023 |
| M.Wt: | 582.65 |
| Formula: | C33H34N4O6 |
| Purity: | >98 % |
| Solubility: | DMSO : ≥ 100 mg/mL |
Azelnidipine (CS 905) is a dihydropyridine calcium channel blocker that is effective orally. Azelnidipine inhibits the intracellular calcium ion flow and lower blood pressure by selectively blocking L-type calcium channel on the membrane of vascular smooth muscle. Azelnidipine inhibits esophageal squamous cell carcinoma proliferation by targeting MEK1/2. Azelnidipine also has anti-inflammatory, antioxidant and neuroprotective effects [1] [2] [3].
In Vitro:Azelnidipine (0-10 μM; 96 h) inhibits esophageal squamous cell carcinoma proliferation by targeting MEK1/2 [2].
In Vivo:Azelnidipine (3 mg/kg/day; Oral gavage; 7 days) plays a protective role in rat models of cerebral ischemia-reperfusion [3].
Azelnidipine (0-3 mg/kg; Oral administration/Intravenous injection; 0-24 h) reduces blood pressure in hypertensive rat models. Oral efficacy is more than three times of Nicardipine (HY-12515). Intravenous injection is three times less effective than Nicardipine (HY-12515) [4].
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