XMD8-87
CAS No. : 1234480-46-6
(Synonyms: ACK1-B19)
| Size | Price | Stock |
|---|---|---|
| 5mg | $90 | In-stock |
| 10mg | $155 | In-stock |
| 25mg | $345 | In-stock |
| 50mg | $525 | In-stock |
| 100mg | $750 | In-stock |
| 200 mg | Get quote | |
| 500 mg | Get quote | |
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| Cat. No. : | HY-15811 |
| M.Wt: | 445.52 |
| Formula: | C24H27N7O2 |
| Purity: | >98 % |
| Solubility: | DMSO : ≥ 26 mg/mL |
XMD8-87 is a potent TNK2 inhibitor with IC50 values of 38 and 113 nM for the D163E and R806Q mutations, respectively. IC50 & Target:IC50: 38 nM (TNK2, D163E mutation), 113 nM (TNK2, R806Q mutation)[1] In Vitro: XMD8-87 potently inhibits the growth of the TNK2 mutant expressing cell lines while having little or no effect on the control cells out to the highest tested concentrations (1,000 nM). XMD8-87 has IC50s of 38 nM and 113 nM for the D163E and R806Q mutations. The effects of XMD8-87 on TNK2 cell lines are largely due to on-target effects on TNK2. Auto-phosphorylation of overexpressed TNK2 mutants could be blocked with TNK2 inhibitor XMD8-87[1].
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