DSP-2230
CAS No. : 1233231-30-5
(Synonyms: ANP-230)
| Size | Price | Stock |
|---|---|---|
| 5mg | $80 | In-stock |
| 10mg | $130 | In-stock |
| 25mg | $280 | In-stock |
| 50mg | $450 | In-stock |
| 100mg | $720 | In-stock |
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| 500 mg | Get quote | |
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| Cat. No. : | HY-125079 |
| M.Wt: | 419.40 |
| Formula: | C20H20F3N5O2 |
| Purity: | >98 % |
| Solubility: | DMSO : ≥ 100 mg/mL |
DSP-2230 is the orally active inhibitor for voltage-gated sodium channel that inhibits Nav1.7-, Nav1.8-, and Nav1.9-derived sodium currents with IC50s of 7.1 μM, 11.4 μM and 6.7 μM, respectively. DSP-2230 can be used to improve neuropathic pain[1][2][3][4]. In Vitro: DSP-2230 inhibits Nav1.7, 1.8, and 1.9 sodium channels, reduces the influx of sodium ions, inhibits the generation and propagation of neuronal action potentials, thereby exhibiting analgesic activity[3]. In Vivo: DSP-2230 (3-30 mg/kg, po, once daily for 6 days) reduces thermal hyperalgesia and mechanical hyperalgesia in R222S mutant mice, inhibits thermal hyperalgesia in wildtype mice[3].
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