KCC2 blocker 1
CAS No. : 1228439-36-8
| Size | Price | Stock |
|---|---|---|
| 5mg | $215 | In-stock |
| 10mg | $315 | In-stock |
| 25mg | $560 | In-stock |
| 50mg | $840 | In-stock |
| 100mg | $1240 | In-stock |
| 200 mg | Get quote | |
| 500 mg | Get quote | |
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| Cat. No. : | HY-18172 |
| M.Wt: | 415.50 |
| Formula: | C22H25NO5S |
| Purity: | >98 % |
| Solubility: | DMSO : 250 mg/mL (ultrasonic) |
KCC2 blocker 1 is an orally active and selective K+-Cl- cotransporter KCC2 blocker with an IC50 of 1 μM. KCC2 blocker 1 is a benzyl prolinate[1].
IC50 & Target:IC50: 1 μM (KCC2)[1]
In Vitro:KCC2 blocker 1 (compound 13; 100 μM) inhibits NKCC1 with 35%.
In Vivo:KCC2 blocker 1 (compound 13; 1 mg/kg iv and 6 mg/kg po) has a t1/2 of 0.3 hours, a CL of 26 mL/min/kg, a C max of 457 ng/mL and a AUC of 726 ng?h/mL for male Wistar rats[1].
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