Naltriben (mesylate)


CAS No. : 122517-78-6

122517-78-6
Price and Availability of CAS No. : 122517-78-6
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5mg $410 In-stock
10mg $750 In-stock
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Cat. No. : HY-101302
M.Wt: 511.59
Formula: C27H29NO7S
Purity: >98 %
Solubility: DMSO : 50 mg/mL (ultrasonic)
Introduction of 122517-78-6 :

Naltriben mesylate is a potent δ2-opioid receptor antagonist and a TRPM7 activator. Naltriben mesylate shows Ki values of 0.013 nM, 19 nM and 152 nM for δ, μ and κ receptors, respectively. Naltriben mesylate enhances glioblastoma cell migration and invasion. Naltriben mesylate can be used in research into neurological diseases and cancer[1][2]. In Vivo:The hypothermia caused by SNC-80 (35 mg/kg, im) is blocked by a delta2 antagonist, Naltriben (2.5 mg/kg; sc; Sprague-Dawley rats weighing 100-125 g)[2].

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