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|---|---|---|
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| 250 mg | Get quote | |
| 500 mg | Get quote | |
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| Cat. No. : | HY-15244R |
| M.Wt: | 441.47 |
| Formula: | C19H22F3N5O2S |
| Purity: | >98 % |
| Solubility: |
Alpelisib (Standard) is the analytical standard of Alpelisib. This product is intended for research and analytical applications. Alpelisib (BYL-719) is a potent, selective, and orally active PI3Kα inhibitor. Alpelisib (BYL-719) shows efficacy in targeting PIK3CA-mutated cancer. Alpelisib (BYL-719) also inhibits p110α/p110γ/p110δ/p110β with IC50s of 5/250/290/1200 nM, respectively. Antineoplastic activity[1][2][3]. IC50 & Target:IC50: 5 nM (p110α), 250 nM (p110γ), 290 nM (p110δ), 1200 nM (p110β)[1]
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