GYKI-47261 (dihydrochloride)
CAS No. : 1217049-32-5
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|---|---|---|
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| 5mg | $1353 | Get quote |
| 10mg | $1960 | Get quote |
| 25mg | $2915 | Get quote |
| 50 mg | Get quote | |
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| Cat. No. : | HY-19435A |
| M.Wt: | 395.71 |
| Formula: | C18H17Cl3N4 |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
GYKI-47261 dihydrochloride is a competitive, orally active, and selective AMPA receptor antagonist with an IC50 of 2.5 μM. GYKI-47261 has broad spectrum anticonvulsive activity and neuroprotective effects. GYKI-47261 dihydrochloride is also a potent inducer of CYP2E1[1][2].
In Vivo: GYKI-47261 dihydrochloride (6 mg/kg; i.v.) shows antiischemice effect in a transient focal ischemia model, in rats. GYKI-47261 dihydrochloride (p.o.) potently mitigated the tremor induced by oxotremorine with ED50 of 16.8 mg/kg in male CD1 mice[1].
GYKI-47261 dihydrochloride(20 mg/kg; i.p.) reverses the dopamine depleting effect of MPTP[1].
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- GYKI-47261 (dihydrochloride)
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