CP 81282
CAS No. : 121584-61-0
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| Cat. No. : | HY-117641 |
| M.Wt: | 635.74 |
| Formula: | C32H47F2N5O6 |
| Purity: | >98 % |
| Solubility: |
CP 81282 is a tripeptide aspartic protease inhibitor containing difluorostatone, with an IC50 of 1 nM against human renin and an IC50 of 11 nM against endopeptidase. CP 81282 is applicable to the research of hypertension[1].
In Vitro:CP 81282 potently inhibits human plasma renin with an IC50 of 1 nM and endothiapepsin with an IC50 of 11 nM[1].
CP 81282 (10-fold molar excess) binds to endothiapepsin as a tetrahedral hydrate, forming specific hydrogen bonds with active-site aspartates 32 and 215, and adopts an extended conformation that interacts with additional enzyme residues[1].
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