Ertugliflozin L-pyroglutamic acid
CAS No. : 1210344-83-4
(Synonyms: PF-04971729 L-pyroglutamic acid)
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|---|---|---|
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| 10mg | $70 | In-stock |
| 50mg | $120 | In-stock |
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| Cat. No. : | HY-15461A |
| M.Wt: | 566.00 |
| Formula: | C27H32ClNO10 |
| Purity: | >98 % |
| Solubility: | DMSO : ≥ 125 mg/mL;H2O : 5 mg/mL (ultrasonic;warming;heat to 60°C) |
Ertugliflozin L-pyroglutamic acid (PF-04971729 L-pyroglutamic acid) is a potent, selective and orally active inhibitor of the sodium-dependent glucose cotransporter 2 (SGLT2), with an IC50 of 0.877 nM for h-SGLT2[1]. Has the potential for the treatment of type 2 diabetes mellitus[2]. IC50 & Target: IC50: 0.877 nM (h-SGLT2)[1]. In Vitro: Ertugliflozin L-pyroglutamic acid (PF-04971729 L-pyroglutamic acid) demonstrates >2000-fold selectivity for SGLT2 inhibition (relative to SGLT1) in vitro[3]. In Vivo: Ertugliflozin L-pyroglutamic acid (PF-04971729 L-pyroglutamic acid) reveals a concentration-dependent glucosuria after oral administration to rats[3].
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