| Size | Price | Stock |
|---|---|---|
| 5mg | $620 | In-stock |
| 10mg | $990 | In-stock |
| 25mg | $1980 | In-stock |
| 50mg | $3170 | In-stock |
| 100 mg | Get quote | |
| 200 mg | Get quote | |
| We match the lowest price on market. | ||
We offer a substantial discount on larger orders, please inquire via [email protected]
or Fax: (86)21-58955996
Inquiry for price and availability only. Please place your order via our email or fax.
| Cat. No. : | HY-106844 |
| M.Wt: | 425.50 |
| Formula: | C22H23N3O4S |
| Purity: | >98 % |
| Solubility: |
EMD 53998 is a cardiotonic agent that increases myocardial contractility as an inhibitor for phosphodiesterase III (PDE III) and a calcium sensitizer. EMD 53998 increases myocardial contractility, reduces energy consumption and the risk of inducing arrhythmias[1]. In Vitro:EMD 53998, a racemic thiadiazinone derivative, is a potent Ca2+-sensitizer. EMD 53998 (0.1-100 μM) increases force of contraction (FOC) in a concentration-dependent manner. EMD 53998 increases force of contraction in human myocardium via sensitizing of the contractile proteins towards Ca2+ and by inhibition of phosphodiesterase III-isoenzymes[12].
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