Delequamine (hydrochloride)
CAS No. : 119942-75-5
(Synonyms: RS-15385-197 (hydrochloride))
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| Cat. No. : | HY-106874A |
| M.Wt: | 386.94 |
| Formula: | C18H27ClN2O3S |
| Purity: | >98 % |
| Solubility: |
Delequamine (RS-15385-197) hydrochloride is an orally active and selective α2-adrenergic receptor antagonist with a pKi of 9.5 for α2-adrenoceptors in rat cortex. Delequamine hydrochloride shows >1000 fold selectivity against 5-HT1A receptors and α1-adrenoceptors. Delequamine hydrochloride can be used for the study of erectile dysfunction[1]. In Vivo:Delequamine (0.4-6.4 mg/kg; oral, single dose) hydrochloride can increase the sexual behavior score in a dose-dependent manner in a model where untrained male rats are exposed to estrogen-progesterone-treated, sexually receptive female rats. Furthermore, the combination of Delequamine (0.4 mg/kg; oral, single dose) hydrochloride and 8-OH-DPAT (HY-112061) (0.1 mg/kg; subcutaneous injection) can increase the percentage of mounts, intromissions, and ejaculations in rats, shorten the ejaculation latency, and reduce the number of intromissions[1].
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