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|---|---|---|
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| Cat. No. : | HY-101685 |
| M.Wt: | 526.62 |
| Formula: | C28H38N4O6 |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
Iganidipine is a Ca2+ antagonist. IC50 & Target: Ca2+[1] In Vivo: Iganidipine (0.03% solution) significantly increases optic nerve head (ONH) tissue blood velocity (NBONH) by 8 to 10% in treated eyes after a single administration (p<0.05) or by 18 to 35% after 7-, 14-, or 21-day twicedaily administration in rabbits (p<0.05). In monkeys, 0.03% and 0.1% Iganidipine significantly increases NBONH in treated eyes by 20 and 41% after 7-day (p<0.05) twice-daily administration, respectively[1].
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