G15
CAS No. : 1161002-05-6
| Size | Price | Stock |
|---|---|---|
| 5mg | $94 | In-stock |
| 10mg | $154 | In-stock |
| 25mg | $290 | In-stock |
| 50mg | $460 | In-stock |
| 100mg | $700 | In-stock |
| 200 mg | Get quote | |
| 500 mg | Get quote | |
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| Cat. No. : | HY-103449 |
| M.Wt: | 370.24 |
| Formula: | C19H16BrNO2 |
| Purity: | >98 % |
| Solubility: | DMSO : 41.67 mg/mL (ultrasonic) |
G15 is a high affinity and selective G-protein-coupled estrogen receptor (GPER/GPR30) antagonist with a Ki of 20 nM[1][2].
IC50 & Target:Ki: 20 nM (GPER/GPR30)[2]
In Vitro: G15 (0.1-10 μM; 2 days) inhibits GPER-mediated proliferation stimulated by 17β-estradiol (E2) in A549 and H1793 cell lines[1].
G15 (1 μM; 48 hours) inhibits the response of GPER stimulated by E2 and G1 in A549 and H1793 cell lines[1].
In Vivo: G15 (1.46 mg/kg; i.h.; twice a week for 14 weeks) decreases the number of tumor nodules and tumor index increased by the E2 or G1 group in urethane-induced adenocarcinoma mice[1].
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