BMS-823778 (hydrochloride)
CAS No. : 1140898-87-8
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| Cat. No. : | HY-120643 |
| M.Wt: | 364.27 |
| Formula: | C18H19Cl2N3O |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
BMS-823778 hydrochloride is a potent, selective and orally active 11β-HSD1 inhibitor with an IC50 of 2.3 nM against human 11β-HSD1[1].
IC50 & Target:IC50: 2.3 nM (human 11β-HSD1), 600 nM (mouse 11β-HSD1)[1]
Ki: 0.9 nM (human 11β-HSD1), 380 nM (mouse 11β-HSD1)[1]
In Vivo: BMS-823778 (10-100 mg/kg; oral; once) hydrochloride exhibits robust acute pharmacodynamic effects in diet-induced obese (DIO) mice (ED50=34 mg/kg) [1].
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