Zaldaride maleate
CAS No. : 109826-27-9
(Synonyms: CGS-9343B; KW 5617)
| Size | Price | Stock |
|---|---|---|
| 1mg | $85 | In-stock |
| 5mg | $210 | In-stock |
| 10mg | $336 | In-stock |
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| Cat. No. : | HY-105118A |
| M.Wt: | 544.60 |
| Formula: | C30H32N4O6 |
| Purity: | >98 % |
| Solubility: | 10 mM in H2O |
Zaldaride maleate (CGS-9343B) is a potent, orally active and selective inhibitor of calmodulin. Zaldaride maleate inhibits CaM (calmodulin)-stimulated cAMP phosphodiesterase activity, with an IC50 of 3.3 nM[1][2]. Zaldaride maleate prevents estrogen-induced transcription activation by ER, reversibly blocks voltage-activated Na+, Ca2+ and K+ currents in PC12 cells and inhibits nAChR[3]. IC50 & Target:IC50: 3.3 nM (calmodulin)[1][2]. In Vivo:Zaldaride (KW 5617, P.O., 3 mg/kg) maleate ameliorates the diarrhea in the 16, 16-dimethyl prostaglandin E2 model[4].
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