Zaldaride
CAS No. : 109826-26-8
(Synonyms: CGS-9343B (free base); KW 5617 (free base))
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| Cat. No. : | HY-105118 |
| M.Wt: | 428.53 |
| Formula: | C26H28N4O2 |
| Purity: | >98 % |
| Solubility: |
Zaldaride (CGS-9343B free base) is a potent, orally active and selective inhibitor of calmodulin. Zaldaride inhibits CaM (calmodulin)-stimulated cAMP phosphodiesterase activity, with an IC50 of 3.3 nM[1][2]. Zaldaride prevents estrogen-induced transcription activation by ER, reversibly blocks voltage-activated Na+, Ca2+ and K+ currents in PC12 cells and inhibits nAChR[3]. IC50 & Target:IC50: 3.3 nM (calmodulin)[1][2]. In Vivo:Zaldaride (P.O., 3 mg/kg) ameliorates the diarrhea in the 16, 16-dimethyl prostaglandin E2 model[4].
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