BI-671800
CAS No. : 1093108-50-9
| Size | Price | Stock |
|---|---|---|
| 1mg | $55 | In-stock |
| 5mg | $135 | In-stock |
| 10mg | $220 | In-stock |
| 25mg | $395 | In-stock |
| 50mg | $560 | In-stock |
| 100mg | $760 | In-stock |
| 200 mg | Get quote | |
| 500 mg | Get quote | |
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| Cat. No. : | HY-114141 |
| M.Wt: | 501.50 |
| Formula: | C25H26F3N5O3 |
| Purity: | >98 % |
| Solubility: | DMSO : 135 mg/mL (ultrasonic) |
BI-671800 is a highly specific and potent antagonist of chemoattractant receptor-homologous molecule on Th2 cells (DP2/CRTH2), with IC50 values of 4.5 nM and 3.7 nM for PGD2 binding to CRTH2 in hCRTH2 and mCRTH2 transfected cells, respectively[1]. BI-671800 has potential for the treatment of poorly controlled asthma[2].
IC50 & Target:CRTH2[1].
In Vitro: BI-671800 (compound A) exhibits low nM potency as an antagonist of human or mouse CRTH2 in transfected cells[1].
In Vivo: BI-671800 (compound A, 0.1-10 mg/kg, i.g.) shows significant inhibition of AHR in mice[1].
BI-671800 (compound A), effectively blocks edema formation and greatly reduces the inflammatory infiltrate and skin pathology observed in drug vehicle-treated animals[3].
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