Protein kinase inhibitor H-7 (dihydrochloride)


CAS No. : 108930-17-2

108930-17-2
Price and Availability of CAS No. : 108930-17-2
Size Price Stock
5mg $55 In-stock
10mg $95 In-stock
25mg $200 In-stock
50mg $320 In-stock
100mg $510 In-stock
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500 mg Get quote
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Cat. No. : HY-100983
M.Wt: 364.29
Formula: C14H19Cl2N3O2S
Purity: >98 %
Solubility: DMSO : 16.67 mg/mL (ultrasonic;warming;heat to 80°C)
Introduction of 108930-17-2 :

Protein kinase inhibitor H-7 dihydrochloride is a potent PKC (protein kinase C) inhibitor. At 100 μM, Protein kinase inhibitor H-7 dihydrochloride completely inhibits both TPA (skin tumour promoter, 12-O-tetradecanoylphorbol-13-acetate) and phospholipase C-induced ODC (ornithine decarboxylase)[1].

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