LDC000067
CAS No. : 1073485-20-7
(Synonyms: LDC067)
| Size | Price | Stock |
|---|---|---|
| 5mg | $54 | In-stock |
| 10mg | $82 | In-stock |
| 25mg | $164 | In-stock |
| 50mg | $246 | In-stock |
| 100mg | $370 | In-stock |
| 200 mg | Get quote | |
| 500 mg | Get quote | |
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| Cat. No. : | HY-15878 |
| M.Wt: | 370.43 |
| Formula: | C18H18N4O3S |
| Purity: | >98 % |
| Solubility: | DMSO : ≥ 47 mg/mL |
LDC000067 is a highly specific CDK9 inhibitor with an IC50 value of 44±10 nM in vitro. IC50 & Target: IC50: 44±10 nM (CDK9-Cyclin T1), 2441 nM (CDK2-Cyclin A)[1] In Vitro: The selectivity of LDC000067 for CDK9 over other CDKs exceeds that of the known inhibitors flavopiridol and DRB. LDC000067 displayed 55/125/210/ >227/ >227-fold selectivity for CDK9 versus CDK2/1/4/6/7. LDC000067 inhibits in vitro transcription in an ATP-competitive and dose-dependent manner. Gene expression profiling of cells treated with LDC000067 demonstrates a selective reduction of short-lived mRNAs, including important regulators of proliferation and apoptosis[1].
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