6-CEPN
CAS No. : 1054549-73-3
| Size | Price | Stock |
|---|---|---|
| 5mg | $500 | In-stock |
| 10mg | $800 | In-stock |
| 25mg | $1600 | In-stock |
| 50 mg | Get quote | |
| 100 mg | Get quote | |
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| Cat. No. : | HY-114569 |
| M.Wt: | 374.39 |
| Formula: | C23H18O5 |
| Purity: | >98 % |
| Solubility: | DMSO : 100 mg/mL (ultrasonic) |
6-CEPN is a RAS inhibitor. 6-CEPN can inhibit RAS activation by binding to Icmt binding sites. 6-CEPN has anticancer activity. 6-CEPN can block cancer cells in the G1 phase. 6-CEPN can induce autophagy and necrosis of Cancer cells (Icmt: isovalerylcysteine carboxymethyltransferase)[1].
IC50 & Target:P21[1].
In Vitro:6-CEPN (10-100 μM, 24 h) decreases cell activity in a dose-dependent manner in SW620, SW480, HCT116 and HT29 cells,and a can resist cell proliferation[1].
6-CEPN (10 μM, 24 h) can block the cell cycle in G1 phase in SW620 and HCT116 cells[1].
6-CEPN (10 μM, 24 h) induces cell necrosis in SW620 and HCT116 cells [1].
6-CEPN (2.5-10 μM, 24 h) induces autophagy and cell death of colon cancer cells by inhibiting RAS activation in SW620 and HCT116 cancer cells[1].
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