ERK-IN-4
CAS No. : 1049738-54-6
| Size | Price | Stock |
|---|---|---|
| 1mg | $50 | In-stock |
| 5mg | $110 | In-stock |
| 10mg | $180 | In-stock |
| 25mg | $378 | In-stock |
| 50mg | $565 | In-stock |
| 100mg | $850 | In-stock |
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| Cat. No. : | HY-113592 |
| M.Wt: | 328.81 |
| Formula: | C14H17ClN2O3S |
| Purity: | >98 % |
| Solubility: | DMSO : 25 mg/mL (ultrasonic;warming;heat to 80°C) |
ERK-IN-4 is an ERK inhibitor binds preferentially to ERK2 with a Kd of 5 μM. ERK-IN-4 specificity inhibits ERK Rsk-1 and Elk-1 phosphorylation. ERK-IN-4 has little effect on ERK protein phosphorylation by its upstream activator MEK1/2[1].
In Vitro:ERK-IN-4 (Compound 76; 10-75 µM; 10 days) completely inhibits cell proliferation, and decreases number of cell colonies[1].
ERK-IN-4 (Compound 76; 100 µM) inhibits ERK-mediated phosphorylation of Rsk-1 on Thr573 and ERK-mediated Elk-1 phosphorylation in HeLa cells[1].
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