Dagrocorat (hydrochloride)
CAS No. : 1044535-61-6
(Synonyms: PF-00251802 (hydrochloride))
| Size | Price | Stock |
|---|---|---|
| 5mg | $850 | In-stock |
| 10mg | $1400 | In-stock |
| 25mg | $2800 | In-stock |
| 50mg | $4500 | In-stock |
| 100mg | $7300 | In-stock |
| 200 mg | Get quote | |
| 500 mg | Get quote | |
| We match the lowest price on market. | ||
We offer a substantial discount on larger orders, please inquire via [email protected]
or Fax: (86)21-58955996
Inquiry for price and availability only. Please place your order via our email or fax.
| Cat. No. : | HY-16718A |
| M.Wt: | 531.01 |
| Formula: | C29H30ClF3N2O2 |
| Purity: | >98 % |
| Solubility: | DMSO : 100 mg/mL (ultrasonic;warming;heat to 60°C) |
Dagrocorat (PF-00251802) hydrochloride is an orally active and selective high-affinity partial agonist of the glucocorticoid receptor. Dagrocorat hydrochloride is also a time-dependent reversible inhibitor of CYP3A (IC50=1.3 μM in human liver microsomes) and CYP2D6 (Ki=0.57 μM in human liver microsomes). Dagrocorat hydrochloride can be used for the research of rheumatoid arthritis[1]. IC50 & Target: IC50: 1.3 μM (CYP3A in human liver microsomes); IC50: 0.57 μM (CYP2D6 in human liver microsomes)[1] In Vitro: Dagrocorat hydrochloride is metabolized by cytochrome P450 (CYP)3A to an N-oxide metabolite. Dagrocorat hydrochloride is a reversible inhibitor of several CYPs, such as CYP3A and CYP2D6[1].
Lorem ipsum dolor sit amet, consectetur adipisicing elit. Autem earum hic iste maiores, nam neque rem suscipit. Adipisci consequatur error exercitationem fugit ipsam optio qui, quibusdam repellendus sed vero! Debitis.
Inquiry Information- Product Name:
- Dagrocorat (hydrochloride)
- Cat. No.:
- HY-16718A
- Quantity:
Your information is safe with us.