Dagrocorat
CAS No. : 1044535-52-5
(Synonyms: PF-00251802)
| Size | Price | Stock |
|---|---|---|
| 1mg | $545 | In-stock |
| 5mg | $850 | In-stock |
| 10mg | $1400 | In-stock |
| 25mg | $2800 | In-stock |
| 50mg | $4500 | In-stock |
| 100mg | $7300 | In-stock |
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| Cat. No. : | HY-16718 |
| M.Wt: | 494.55 |
| Formula: | C29H29F3N2O2 |
| Purity: | >98 % |
| Solubility: | DMSO : 250 mg/mL (ultrasonic) |
Dagrocorat (PF-00251802) is an orally active and selective high-affinity partial agonist of the glucocorticoid receptor. Dagrocorat is also a time-dependent reversible inhibitor of CYP3A (IC50=1.3 μM in human liver microsomes) and CYP2D6 (Ki=0.57 μM in human liver microsomes). Dagrocorat can be used for the research of rheumatoid arthritis[1]. IC50 & Target: IC50: 1.3 μM (CYP3A in human liver microsomes); IC50: 0.57 μM (CYP2D6 in human liver microsomes)[1] In Vitro: Dagrocorat is metabolized by cytochrome P450 (CYP)3A to an N-oxide metabolite. Dagrocorat is a reversible inhibitor of several CYPs, such as CYP3A and CYP2D6[1].
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