CGP 25454A
CAS No. : 104391-26-6
| Size | Price | Stock |
|---|---|---|
| 5mg | $280 | In-stock |
| 10mg | $480 | In-stock |
| 25mg | $720 | In-stock |
| 50mg | $960 | In-stock |
| 100mg | $1650 | In-stock |
| 200 mg | Get quote | |
| 500 mg | Get quote | |
| We match the lowest price on market. | ||
We offer a substantial discount on larger orders, please inquire via [email protected]
or Fax: (86)21-58955996
Inquiry for price and availability only. Please place your order via our email or fax.
| Cat. No. : | HY-100454 |
| M.Wt: | 346.25 |
| Formula: | C15H21Cl2N3O2 |
| Purity: | >98 % |
| Solubility: | DMSO : ≥ 3.5 mg/mL |
CGP 25454A is a selective presynaptic dopamine autoreceptor antagonist which induces the increase of dopamine and acetyl choline. CGP 25454A can be used for major depression research[1].
In Vitro:CGP 25454A (0.5-10 μM, 15 min) elicits a reproducible and concentration-dependent increase of the release of both DA and ACh in rat striatal slices with an increase by 62±3% and 100±7% at 10 μM. CGP 25454A is 12.9 fold more potent at pre- than post-synaptic DA receptors[1].
In Vivo:CGP 25454A (10-100 mg/kg, i.p., 60 min) produces a marked, close-dependent increase in Spiperone binding in rat striatum[1].
CGP 25454A (0.5-100 mg/kg, i.p., 10-60 min) exerts opposite effects with a slight behavioral stimulation at low doses and a clear-cut central depressant action in the higher dose range[1].
Lorem ipsum dolor sit amet, consectetur adipisicing elit. Autem earum hic iste maiores, nam neque rem suscipit. Adipisci consequatur error exercitationem fugit ipsam optio qui, quibusdam repellendus sed vero! Debitis.
Inquiry Information- Product Name:
- CGP 25454A
- Cat. No.:
- HY-100454
- Quantity:
Your information is safe with us.