MCH-1 antagonist 1
CAS No. : 1039825-68-7
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| Cat. No. : | HY-100331 |
| M.Wt: | 414.50 |
| Formula: | C25H26N4O2 |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
MCH-1 antagonist 1 is a potent melanin concentrating hormone (MCH-1) antagonist with a Ki of 2.6 nM. MCH-1 antagonist 1 also inhibits CYP3A4 with an IC50 of 10 μM.
IC50 & Target: Ki: 2.6 nM (MCH-1)[1]
IC50: 10 μM (CYP3A4)[1]
In Vitro: MCH-1 antagonist 1 (Compound 1) also inhibits cytochrome P450 3A4 (CYP3A4) with an IC50 of 10 μM[1].
In Vivo: MCH-1 antagonist 1 is administered to male C57BL/6J DIO mice to assess their pharmacokinetic profile. Effect of MCH-1 antagonist 1 (dosed at 30 mg/kg, po) is measured on the body weight of DIO mice with the AUC0-6 h of 14760 h*ng/mL[1].
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