Urotensin-II receptor antagonist-1
CAS No. : 1034708-07-0
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| Cat. No. : | HY-10672 |
| M.Wt: | 460.44 |
| Formula: | C25H31Cl2N3O |
| Purity: | >98 % |
| Solubility: |
Urotensin-II receptor antagonist-1 (compound 1) is a low oral bioavailability (F=0-3%, rat) selective human Urotensin II receptor antagonist, Ki=16 nM (test on HEK293 cells expressing recombinant human UT receptor). Urotensin-II receptor antagonist-1 inhibits cytochrome P450 (IC50=0.75 μM, CYP2D6; 1.4 μM, CYP3A4), inhibits κ-opioid receptor (EC50=3.2 μM), targets cardiac sodium channels (Ki=2.5 μM)[1]. IC50 & Target:Urotensin II, κ-Opioid Receptor[1]
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- Cat. No.:
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