Artefenomel
CAS No. : 1029939-86-3
(Synonyms: OZ439)
| Size | Price | Stock |
|---|---|---|
| 1mg | $200 | In-stock |
| 5mg | $450 | In-stock |
| 10mg | $750 | In-stock |
| 25mg | $1400 | In-stock |
| 50mg | $2250 | In-stock |
| 100mg | $3350 | In-stock |
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| Cat. No. : | HY-16762 |
| M.Wt: | 469.61 |
| Formula: | C28H39NO5 |
| Purity: | >98 % |
| Solubility: | DMSO : 4.2 mg/mL (ultrasonic) |
Artefenomel (OZ439) is an orally active, synthetic anti-malarial compound containing an artemisinin pharmacophore with a mechanism of action similar to that of artemisinin. Artefenomel has antiviral activity against SARS-CoV-2[1][2].
In Vitro: Artefenomel (OZ439) (10 μg/mL, 2 h) can alkylate Plasmodium falciparum proteins[1].
Artefenomel (0.3-300 μM) reduces ACE2 expression in Vero cells in a dose-dependent manner and does not induce any cytotoxicity at concentrations up to 300 μM[2].
Artefenomel (33-100 μM) can completely prevent the virus-induced CPE and inhibit SARS-CoV-2 in a dose-dependent manner with an IC50 of 2.9 µM[2].
Artefenomel (0-10 µg/mL) affects red blood cells and induces anaemia, thereby inducing histological changes (cell death) and macroscopic abnormalities in the embryo from pregnant Crl:CD(SD)BR rats[3].
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