CB1 inverse agonist 2
CAS No. : 1019839-52-1
| Size | Price | Stock |
|---|---|---|
| 5mg | $210 | In-stock |
| 10mg | $340 | In-stock |
| 25mg | $688 | In-stock |
| 50mg | $1100 | In-stock |
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| Cat. No. : | HY-12095 |
| M.Wt: | 438.94 |
| Formula: | C24H20ClFN2OS |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
CB1 inverse agonist 2 is an orally active inverse agonist of Cannabinoid Receptor CB1. CB1 inverse agonist 2 effectively inhibits CP55940-induced hypothermia and anorexia in mice model[1].
In Vitro:CB1 inverse agonist 2 (compound 12 h) shows selectivity on CB1 over CB2 with pKi values of 9.7 and 6.0, respectively[1].
In Vivo:CB1 inverse agonist 2 (compound 12 h) (1 mg/kg; i.p.; single dose) results 70% inhibition against hypothermia, as well as (10 mg/kg; p.o.; single dose) resulting 59% inhibition against food intake[1].
CB1 inverse agonist 2 (10 mg/kg; p.o.; once daily for 14 d) produces robust weight loss of approximately 13% of initial body weight in mouse[1].
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