CVT-10216
CAS No. : 1005334-57-5
| Size | Price | Stock |
|---|---|---|
| 5mg | $125 | In-stock |
| 10mg | $215 | In-stock |
| 25mg | $430 | In-stock |
| 50mg | $688 | In-stock |
| 100 mg | Get quote | |
| 200 mg | Get quote | |
| We match the lowest price on market. | ||
We offer a substantial discount on larger orders, please inquire via [email protected]
or Fax: (86)21-58955996
Inquiry for price and availability only. Please place your order via our email or fax.
| Cat. No. : | HY-19801 |
| M.Wt: | 465.48 |
| Formula: | C24H19NO7S |
| Purity: | >98 % |
| Solubility: | DMSO : 20 mg/mL (ultrasonic;warming);DMF : 25 mg/mL (ultrasonic;warming) |
CVT-10216 is a highly selective, reversible aldehyde dehydrogenase-2 (ALDH-2) inhibitor with an IC50 of 29 nM. CVT-10216 also has inhibitory effect of ALDH-1 with an IC50 of 1.3 μM. CVT-10216 can reduce excessive alcohol drinking in alcohol-preferring rats and exhibit anxiolytic effects[1]. IC50 & Target: IC50: 29 nM (ALDH-2)[1] In Vivo: CVT-10216 (intraperitoneal?injection; 3.75, 7.5, or 15 mg/kg) exhibits a increase in social interaction as a dose-dependent manner, punctuated by a 2-fold increase in social interaction after 15 mg/kg in Fawn-Hooded rats[1]. CVT-10216 (intraperitoneal?injection; 3.75 or 15 mg/kg) are determined 5 h into the third withdrawal.It has the anxiolytic effect of 15 mg/kg CVT-10216 in this model, but has no significant effects on locomotor activity[1].
Lorem ipsum dolor sit amet, consectetur adipisicing elit. Autem earum hic iste maiores, nam neque rem suscipit. Adipisci consequatur error exercitationem fugit ipsam optio qui, quibusdam repellendus sed vero! Debitis.
Inquiry Information- Product Name:
- CVT-10216
- Cat. No.:
- HY-19801
- Quantity:
Your information is safe with us.